December 5-7, 2016 Dubai, UAE

International Conference onMedicinal and Pharmaceutical Chemistry

PharmaMed-2016

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Day 1 - December 5, 2016 - Al Shaheen08:00-09:30 Registrations

09:30-10:00 Opening Ceremony

Keynote Forum

10:00-10:30Title: Key requirements for successful transnational drug discovery projects

Sheraz Gul, Fraunhofer Institute for Molecular Biology & Applied Ecology, Germany

10:30-11:00Title: Applications in pharmaceuticals and drug analysis of modifi ed carbon paste electrodes using different voltammetric techniques

Mahmoud Khodari, South Valley University, Egypt

Coffee Break: 11:00-11:15 @ Foyer B

Session 1: Novel Opportunities for Drug Discovery and Medicinal ChemistrySession Chairs: Raphael Stoll, Ruhr University of Bochum, Germany Rebamang A. Mosa, University of Zululand, Republic of South Africa

11:15-11:40Title: Ruthenium-conjugated synthetic fl avonoid derivatives as novel modulators of platelet function

Sakthivel Vaiyapuri, University of Reading, UK

11:40-12:05Title: Lead modifi cation approaches in the design, synthesis and evaluation of novel chemical entities for muscarinic acetylcholine receptors

Richie R. Bhandare, Ajman University of Science and Technology, UAE

12:05-12:30Title: Biological activity of nanocomposites consisting of TiO2 nanoparticles and antisense oligonucleotides

Asya S. Levina, Novosibirsk State University, Russia

12:30-12:55Title: Bisphenol an analogues bind to ras proteins and compete with guanine nucleotide exchange

Raphael Stoll, Ruhr University of Bochum, Germany

Lunch Break: 12:55-14:00 @ Restaurant

14:00-14:25Title: Toward the design of novel antimicrobials: Synthesis and biological evaluation of phosphate isosters of fosmidomycin and analogs

Catherine Grosdemange-Billiard, Université de Strasbourg/CNRS, France

14:25-14:50Title: Cardioprotective potential of a lanosteryltriterpene from Protorhuslongifolia

Rebamang A. Mosa, University of Zululand, Republic of South Africa

14:50-15:15Title: Structural modifi cations of kidney cystatin in renal cancers

Mohd Anas Shamsi, Aligarh Muslim University, India

15:15-15:40Title: The dual-acting AChEInhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced byscopolamine or dizocilpinein passive avoidance paradigm in rats

Bassem Sadek, United Arab Emirates University, United Arab Emirates

15:40-16:05Title: Physicochemical analysis of antioxidant compounds in fresh juice from cactus cladodes

TALBI Meryeme, University Hassan 1er, Morocco

Coffee Break: 16:05-16:20 @ Foyer B

Day 2 - December 6, 2016 - Al ShaheenKeynote Forum

09:30-10:00Title: Biomolecular NMR spectroscopy in medicinal chemistry

Raphael Stoll, Ruhr University of Bochum, Germany

10:00-10:30Title: Protective effects of apricot againist ketamin ıncuduced hepatotoxicity in rats

Ismet Yilmaz, Inonu University, Turkey

Coffee Break: 10:30-10:45 @ Foyer B

Session 2: Antibiotics and Anti Cancer Drugs Molecular Modeling and Computer-Aided Drug Design Pharmaceutical Analysis: Analytical MethodsSession Chairs: Mahmoud Khodari, South Valley University, Egypt

10:45-11:10Title: Fluoroquinolone-associated toxicities: Tipping the risk-benefi t scale

Monique R. Bidell, Albany College of Pharmacy and Health Sciences, USA

11:10-11:35Title: Design, synthesis and biological characterization of chalcones and propanediones as inhibitors of histone methyl transferase against leukemia cell lines

C. S Ramaa, Bharati Vidyapeeth’s College of Pharmacy, India

11:35-12:00Title: Discovery and optimization of novel antagonists of the WDR5-MLL interaction

Rima Al-awar, University of Toronto, Canada

12:00-12:25Title: Homology modelling, structure- and ligand-based drug design of novel tubulin inhibitors and calcium channel blockers with anti- proliferative and leishmanicidal activities

Carlos Henrique Tomich de Paula da Silva, University of São Paulo, Brazil

12:25-12:50Title: Selective electrochemical determination of desipramine using a lipid modifi ed carbon paste electrode

Mahmoud Khodari, South Valley University, Egypt

Lunch Break: 12:50-13:35 @ Restaurant

Session 3: Drug Design, Discovery and Development Pharmaceutical Analysis: Analytical Methods Pharmacology and ToxicologySession Chairs: Usharani Pingali, Nizam’s Institute of Medical Sciences (NIMS), India Marcela Krečmerová, Czech Academy of Sciences, Czech Republic

13:35-14:00Title: Antiviral acyclic nucleoside phosphonates: New structures and prodrugs

Marcela Krečmerová, Czech Academy of Sciences, Czech Republic

14:00-14:25Title: Design and synthesis of benzoazoles incorporating fl uorine and piperazine moieties with potential biological activities

Raid Abdel-jalil, Sultan Qaboos University, Oman

14:25-14:50Title: A Study of highly standardized aqueous extract of Terminalia chebula 250mg, 500mg versus Placebo in modifying cardiovascular risk with special reference to Endothelial dysfunction in patients with Type2 Diabetes

Usharani Pingali, Nizam’s Institute of Medical Sciences (NIMS), India

14:50-15:15Title: Structure-affi nity and structure-kinetics relationship study: A new combination strategy in medicinal chemistry

Dong Guo, Xuzhou Medical University, China

15:15-15:40Title: Synthesis, anti-inflammatory, analgesic, molecular modeling and admet studies of diclofenylalanylhydrazide

Magda Hassan Abd El Lattif, Taif University, Kingdom of Saudi Arabia

15:40-16:05Title: Synthesis of zinc oxide doped- poly(8-anilino-1-napthlene sulphonic acid) (ZnO/PANSA) as conducting platforms for TB drug biosensors

Rachel Ajayi, University of the Western Cape, South Africa

Coffee Break: 16:05-16:15 @ Foyer B

Workshop

16:15-18:00Title: A critical evaluation of assays in pre-clinical drug discovery

Sheraz Gul, Fraunhofer Institute for Molecular Biology & Applied Ecology, Germany

Day 3 - December 7, 2016 - Al ShaheenPoster Presentations: 10:00-12:30 @ Foyer B

P1Title: Role of formyl peptide receptors in the regulation of thrombosis and haemostasis

Maryam Salamah, University of Reading, UK

P2Title: Cytotoxic effects of bioactive compounds isolated of Iris persica L. on human cancer cell lines

Faiq H. S. Hussain, University of Salahaddin, Iraq

P3Title: A practical and eco-friendly synthesis of oxo-bile acids

Hwayoung Yun, Pusan National University, Republic of Korea

P4Title: Synthesis and cellular uptake of nanocomposites containing oligonucleotides and their analogues immobilized on inorganic nanoparticles

Marina N. Repkova, Novosibirsk State University, Russia

P5Title: In-vitro antidiabetic activity of partially purifi ed fractions of Pithecellobium dulce fruit

Preethi S, VIT University, India

P6Title: Apoptosis versus autophagy in the molecular mechanism of action of plant derived chemotherapeutics against hepatocellular carcinoma cells

Greeshma Tom, Rajiv Gandhi Centre for Biotechnology, India

P7Title: Anti-infl ammatory action through inhibition of NF kB activation and translocation by band-2 isolated from Tinospora cordifolia(Thunb.) miers. in LPS stimulated RAW 264.7 cell lines

Sheena Philip, Rajiv Gandhi Centre for Biotechnology, India

P8Title: Identifi cation of structural elements of MCP chemokines and their shared receptor CCR2

Zil e Huma, Monash University, Australia

P9Title: Targeting bacterial stringent response

Dominik Rejman, Czech Academy of Sciences v.v.i., Czech Republic

P10Title: Characterization of nucleotide pool in bacterial cells

Eva Zborníková, Czech Academy of Sciences v.v.i., Czech Republic

P11Title: Design TiO2 nanoparticles for using in nanocomposites containing oligonucleotides and their analogues

Elena V Bessudnova, Novosibirsk State University, Russia

P12Title: Low dose irbesartan has a renoprotective effect as high dose ramipril in diabetic rats treated with insulin

Abdulelah A. Thigah, Umm Al-Qura university, Saudi Arabia

P13Title: Aspirin and blood glucose and insulin resistance

Abdullah A. Alshamrani, Umm Al-Qura university, Saudi Arabia

P14Title: Prevalence and preventive measures of infertility in male by kruger’s criteria, a randomized study in private and government health care hospitals

Huda Ashraf, Jinnah University for Women, Pakistan

P15Title: In silico pharmacokinetics and molecular docking of three leads isolated from Tarconanthus Camphoratus L

Amina I. Dirar, Medicinal and Aromatic Plants Research Institute, Sudan

P16Title: Zika virus NS5 protein potential inhibitors: An enhanced in silico approach in drug discovery

Pritika Ramharack, University of KwaZulu-Natal, South Africa

Coffee Break: 11:00-11:15 @ Foyer B

Award Ceremony